4SC-202 |
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(CAS 1186222-89-8) |
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Description: |
4SC-202 is an orally available potent HDACi specific for class I HDAC isoenzymes(NO HDAC8) with IC50s of 1.2/1.12/0.57 uM for HDAC1/2/3; high selectivity over ClassIIa/IIb/III HDACs.
The novel HDACi 4SC-202 is an orally available potent HDACi specific for class I HDAC isoenzymes. It has shown substantial anti-tumour activity in a broad panel of cancer cell lines as well as in various cancer xenograft models. A Phase I study with 4SC-202 in haematological malignancies is currently prepared and about to start soon. |
Product No. |
KT01028 |
Product Name |
4SC-202 |
Synonyms |
4SC 202; 4SC202 |
Formal Name |
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CAS Number |
1186222-89-8 |
Molecular Formula |
C30H29N5O6S2 |
Formula Weight |
619.71 |
Formulation |
A crystalline solid |
Purity |
98%min |
Stability |
2 years |
Storage |
-20°C |
Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
Price & Availability |
In Stock. Price Negotiated. |
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