| GSK1070916 |
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| (CAS 942918-07-2) |
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| Description： |
GSK1070916 selectively inhibits Aurora B and Aurora C with Ki of 0.38 nM and 1.5 nM over Aurora A with Ki of 490 nM. Inhibition of Aurora B and Aurora C is time-dependent, with an enzyme-inhibitor dissociation half-life of >480 min and 270 min respectively. In addition, GSK1070916 is also a competitive inhibitor with respect to ATP.
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| Product No. |
KT00389 |
| Product Name |
GSK1070916 |
| Synonyms |
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| Formal Name |
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| CAS Number |
942918-07-2 |
| Molecular Formula |
C30H33N7O |
| Formula Weight |
507.63 |
| Formulation |
A crystalline solid |
| Purity |
98%min |
| Stability |
2 years |
| Storage |
-20°C |
| Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
| Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
| Price & Availability |
In Stock. Price Negotiated. |
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| Related Products： |
Alisertib
AMG 900
AT9283
Aurora A inhibitor I
AZD1152
AZD1152-HQPA
CCT 137690
CCT129202
CYC-116
ENMD-2076
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