BRL54443 |
3-(1-methylpiperidin-4-yl)-1H-indol-5-ol |
(CAS 57477-39-1) |
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Description: |
BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively); displays > 30-fold selectivity over other 5-HT and dopamine receptors.
in vivo: Reduction of flinching was considered as antinociception. Ipsilateral, but not contralateral, peripheral administration of BRL54443 (5-HT(1E/1F); 3-300 microg/paw) significantly reduced formalin-induced flinching in rats [3].
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Product No. |
KT00226 |
Product Name |
BRL54443 |
Synonyms |
BRL54443 |
Formal Name |
3-(1-methylpiperidin-4-yl)-1H-indol-5-ol |
CAS Number |
57477-39-1 |
Molecular Formula |
C14H18N2O |
Formula Weight |
230.31 |
Formulation |
A crystalline solid |
Purity |
98%min |
Stability |
2 years |
Storage |
-20°C |
Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
Price & Availability |
In Stock. Price Negotiated. |
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