| BTS54524 |
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| (CAS 84485-00-7) |
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| Description： |
Sibutramine Hydrochloride(BTS 54-524) is a serotonin and noradrenaline reuptake inhibitor.
Target: SSRIs
Sibutramine is a novel 5-HT (serotonin) and noradrenaline reuptake inhibitor (SNRI) anti-obesity drug. Sibutramine is an oral anorexiant. Sibutramine is a neurotransmitter reuptake inhibitor that reduces the reuptake of serotonin (by 53%), norepinephrine (by 54%), and dopamine (by 16%), thereby increasing the levels of these substances in synaptic clefts and helping enhance satiety; the serotonergic action, in particular, is thought to influence appetite. Older anorectic agents such as amphetamine and fenfluramine force the release of these neurotransmitters rather than affecting their reuptake [1].
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| Product No. |
KT20769 |
| Product Name |
BTS54524 |
| Synonyms |
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| Formal Name |
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| CAS Number |
84485-00-7 |
| Molecular Formula |
C17H27Cl2N |
| Formula Weight |
316.31 |
| Formulation |
A crystalline solid |
| Purity |
98%min |
| Stability |
2 years |
| Storage |
-20°C |
| Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
| Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
| Price & Availability |
In Stock. Price Negotiated. |
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| Related Products： |
Azaphen
Pipofezine(Azafen or Azaphen) is a potent inhibitor of the reuptake of serotonin.
IC50 Value:
Target: SSRIs
Pipofezine is a tricyclic antidepressant (TCA) approved in Russia for the treatment of depression. In addition to its antidepressant action, pipofezine has sedative effects as well, indicating antihistamine activity.
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