WIN54461 |
[6-bromo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone |
(CAS 166599-63-9) |
 |
Description: |
WIN54461 is an aminoalikylindole which acts as a cannabinoid (CB) mimetic, displacing WIN 55212-2 from CB receptors on rat cerebellum membranes (IC50 = 515 nM).As it antagonizes the inhibition of electrically-induced contractions in isolated mouse vas deferens preparations by tetrahydrocannabinol or pravadoline, it may act as a receptor antagonist.The physiological effects of WIN54461 in vivo have not been examined. This product is intended for research and forensic applications.
|
Product No. |
KT00735 |
Product Name |
WIN54461 |
Synonyms |
6-Bromopravadoline |
Formal Name |
[6-bromo-2-methyl-1-[2-(4-morpholinyl)ethyl]-1H-indol-3-yl](4-methoxyphenyl)-methanone |
CAS Number |
166599-63-9 |
Molecular Formula |
C23H25BrN2O3 |
Formula Weight |
457.36 |
Formulation |
A crystalline solid |
Purity |
98%min |
Stability |
2 years |
Storage |
-20°C |
Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
Price & Availability |
In Stock. Price Negotiated. |
|
Related Products: |
WIN18446
(+)-WIN 55,212-2 (mesylate)
(−)-WIN 55,212-3 (mesylate)
(±)-WIN 55,212 (mesylate)
|
|