Talipexole dihydrochloride |
6-Allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepine-2-amine dihydrochloride |
(CAS 36085-73-1) |
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Description: |
B-HT 920(Talipexole 2Hcl) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist and 5-HT3 receptor antagonist, which displays antiParkinsonian activity.
IC50 Value: 25 nM(Adrenergic receptor α-2, rat)
Target: Adrenergic Receptor; 5-HT Receptor; Dopamine Receptor
in vitro: N/A
in vivo: Intravenous injection of 30 micrograms/kg of B-HT 920 into cats lead initially to an increase in blood pressure and then to a long-lasting decrease in blood pressure and heart rate. Vagally mediated reflex bradycardia elicited by angiotensin injection in beta-adrenoceptor-blocked dogs was facilitated by intracisternal injection of 10 micrograms/kg B-HT 920.
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Product No. |
KT20226 |
Product Name |
Talipexole dihydrochloride |
Synonyms |
Domin; Talipexole dihydrochloride |
Formal Name |
6-Allyl-5,6,7,8-tetrahydro-4H-thiazolo[4,5-d]azepine-2-amine dihydrochloride |
CAS Number |
36085-73-1 |
Molecular Formula |
C10H15N3S.2(HCl) |
Formula Weight |
282.24 |
Formulation |
A crystalline solid |
Purity |
98%min |
Stability |
2 years |
Storage |
-20°C |
Shipping |
USD45 for Europe and USA. No shipping charge once amount reach USD500 |
Quality Control |
HNMR,CNMR,LCMS,HPLC,IR,etc. |
Price & Availability |
In Stock. Price Negotiated. |
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